Drug misuse

 

Psychotropic drugs are taken as a result of positive reinforcement, e.g. alcohol, cocaine, opium, nicotine, eating and sex all increase dopamine activity.

 

Dependence – a pattern of repeated self –administration that usually results in tolerance, withdrawal and compulsive drug taking behaviour.

 

 

Nicotine

Causes stress, tension, depression and irritability

Smokers feel normal with nicotine but abnormal without it

Nicotine binds to acetylcholine receptors in the PNS and CNS

Causes increased activity of dopamine, noradrenaline, glutamate and serotonin

Increases heart rate by 10 beats per minute via sympathetic effects, so may increase BP and cardiac distress directly.

 

 

Alcohol

 

Types of drinker

1. Social

2. Problem drinker, this will lead to physical, psychological or social harm

3. Heavy drinker, medically unsafe in the long term

4. Binge drinkers, people who drink excessively over a period up to 48 hours

5. Alcohol dependent drinkers, have a physical dependence on alcohol, `alcohol dependency syndrome`.

 

Delirium tremens (DTs)

Occurs 1 – 3 days after alcohol cessation.

Features

Disorientated, agitated, tremor, hallucinations, sweating, tachycardia, tachypnoea, pyrexia

Complications

Dehydration, infections, hepatic disease, Wernick-Korsakoff syndrome

 

 

Solvents

Have an intoxicating effect

Death may occur through asphyxiation or acute poisoning

 

 

Amfetamines

Stimulate the release of monoamines from presynaptic neurone, so act as an indirect agonist

Cause stimulation and euphoria followed by fatigue and depression.

Acute paranoid psychosis may develop, same as acute paranoid schizophrenia

 

 

 

 

 

 

Ecstasy

3, 4-methylenedioxy-methamfetamine (MDMA) is an amphetamine derivative

Psychodelic dance or rave drug, acts for 4-6 hours

Ongoing use can cause neurotransmitter changes in the brain

Can cause malignant hyperpyrexia and dehydration.

Acute renal or hepatic failure are possible.

 

 

Cocaine

CNS stimulant with similar effects to amfetamines

Derived from South American coca trees

Free base or `crack` cocaine can be smoked

Increases dopamine activity

 

 

Hallucinogenic drugs

Lysergic acid diethylamide, mescaline, psilocybin

Frank hallucinations with possible long term psychosis.

Bind to serotonin receptors

 

 

Cannabis

Exaggerates the pre-existing mood

Leeds to tolerance and dependence

Some analgesic and antiemetic properties

Regular use leads to an amotivational syndrome

Cannabis binds to a specific CNS receptor

 

 

Tranquillizers

Benzodiazepines and barbiturates

Benzodiazepines increase GABA activity

Rebound effects may occur

 

 

Opiates

Physical dependence occurs with opium, morphine codeine and heroin

Also occurs with synthetic compounds such as methadone and pethidine

Opiates bind to endorphin receptors

Tolerance is marked

Associated with complications of injecting

Have a severe withdrawal syndrome, worst after 2 – 3 days but recovery occurs after a week.